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Immunotherapy

CTLA-4 Inhibitor

Also known as: Anti-CTLA-4 therapy, CTLA-4 blockade

Definition

A checkpoint inhibitor that blocks CTLA-4 protein, enhancing early T-cell activation against cancer.

Detailed Explanation

CTLA-4 (Cytotoxic T-Lymphocyte Antigen-4) inhibitors work earlier in the immune response than PD-1 inhibitors. Ipilimumab (Yervoy) is the main CTLA-4 inhibitor, often combined with PD-1 inhibitors for better efficacy. It has more immune-related side effects than PD-1/PD-L1 inhibitors but can produce durable responses.